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 About 16 results found for searched term "IOX4" (0.055 seconds)

Cat.No.  Name Target
M11006 IOX4 HIF
IOX4 is a selective PHD2 inhibitor,IC50 With a value of 1.6 nM, HIFα expression is induced in cells and wild-type mice to permeate the blood-brain barrier. IOX4 competes with and displaces 2-oxoglutaric acid (2OG) at the PHD2 active site.
M16349 9β,13β-Epidioxyabiet-8(14)-en-18-oic acid Diterpenoids
9β,13β-Epidioxyabiet-8(14)-en-18-oic acid
M16895 2,3-Di(3',4'-methylenedioxybenzyl) -2-buten-4-olide Lignans
2,3-Di(3',4'-methylenedioxybenzyl) -2-buten-4-olide
M16993 2-(2,2-Dimethyl-1,3-dioxolan -4-yl)propane-1,2-diol Others
2-(2,2-Dimethyl-1,3-dioxolan -4-yl)propane-1,2-diol
M16994 1,6-Dioxaspiro[4.5]decan-2-methanol Others
1,6-Dioxaspiro[4.5]decan-2-methanol
M43876 1,1-Dimethylethyl 6-(2,6-dioxo-3-piperidinyl)-3,4-dihydro-2(1H)-isoquinolinecarboxylate Ligand for E3 Ligase
1,1-Dimethylethyl 6-(2,6-dioxo-3-piperidinyl)-3,4-dihydro-2(1H)-isoquinolinecarboxylate
M41897 RTIOXA-43 OX Receptor
RTIOXA-43 is a orexin receptor agonist with EC50s of 24 nM and 24 nM for OX2 and OX1 receptors, respectively.
M43847 1-(4-(2,6-dioxopiperidin-3-yl)phenyl)piperidine-4-carbaldehyde Ligand for E3 Ligase
4-Piperidinecarboxaldehyde, 1-[4-(2,6-dioxo-3-piperidinyl)phenyl]-
1-(4-(2,6-dioxopiperidin-3-yl)phenyl)piperidine-4-carbaldehyde
M43851 1-[5-(2,6-Dioxo-3-piperidinyl)-2-pyridinyl]-4-piperidineacetic acid Ligand for E3 Ligase
1-[5-(2,6-Dioxo-3-piperidinyl)-2-pyridinyl]-4-piperidineacetic acid
M43860 1-[5-(2,6-Dioxo-3-piperidinyl)-3-fluoro-2-pyridinyl]-4-piperidineacetic acid Ligand for E3 Ligase
1-[5-(2,6-Dioxo-3-piperidinyl)-3-fluoro-2-pyridinyl]-4-piperidineacetic acid
M43875 2(1H)-Isoquinolineacetic acid, 6-(2,6-dioxo-3-piperidinyl)-3,4-dihydro- Ligand for E3 Ligase
2(1H)-Isoquinolineacetic acid, 6-(2,6-dioxo-3-piperidinyl)-3,4-dihydro-
M43882 1-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)phenyl)piperidine-4-carbaldehyde Ligand for E3 Ligase
4-Piperidinecarboxaldehyde, 1-[4-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-
1-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)phenyl)piperidine-4-carbaldehyde
M43884 1-[4-(Tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-4-piperidinecarboxylic acid Ligand for E3 Ligase
1-[4-(Tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-4-piperidinecarboxylic acid
M43887 1-(5-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)pyridin-2-yl)piperidine-4-carbaldehyde Ligand for E3 Ligase
4-Piperidinecarboxaldehyde, 1-[5-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)-2-pyridinyl]-
1-(5-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)pyridin-2-yl)piperidine-4-carbaldehyde
M43892 3-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)-4-fluorobenzoic acid Ligand for E3 Ligase
Benzoic acid, 4-fluoro-3-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)-
3-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)-4-fluorobenzoic acid
M44596 11alpha-hydroxy-3,7-dioxo-5alpha-lanosta-8,24(E)-dien-26-oic acid Others
11alpha-hydroxy-3,7-dioxo-5alpha-lanosta-8,24(E)-dien-26-oic acid



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